Optimization of Preparation Technology for -Asarone Cataplasm
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Optimization of Preparation Technology for -Asarone Cataplasm
Chinese Journal of Experimental Traditional Medical FormulaeVol. 18, Issue 6, Pages: 42-45(2012)
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Published:2012
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LIU Lin, FANG Yong-qi, XUE Zhong-feng, et al. Optimization of Preparation Technology for -Asarone Cataplasm[J]. Chinese journal of experimental traditional medical formulae, 2012, 18(6): 42-45.
DOI:
LIU Lin, FANG Yong-qi, XUE Zhong-feng, et al. Optimization of Preparation Technology for -Asarone Cataplasm[J]. Chinese journal of experimental traditional medical formulae, 2012, 18(6): 42-45.DOI:
Optimization of Preparation Technology for -Asarone Cataplasm
Objective: To optimize preparation process of β-asarone cataplasm. Method: Orthogonal design test was employed to optimize matrix proportion and molding technology of β-asarone cataplasma with glossiness
adhesiveness
matrix residue
skin following and repeatedly exposing as indexes. Result: Optimum matrix proportion of carbomer-pressure sensitive adhesive-polyvinyl alcohol-sodium carboxymethy cellulose-gelatinum-citric acid-sodium citrate-glycerol-propylene glycol was 0.3:1:0.05:0.35:0.1:0.12:0.18: 3.5:3.5. Optimized molding technology were that stiring speed was 500 r·min-1
refining temperature was 45 ℃
refining time was 15 min
the content of of β-asarone was 8.7%. Conclusion: Optimized β-asarone cataplasm had a good adhesive power
excipients and glossiness
drug loading was large and no skin left.This preparation had a certain advantages and wide application prospects for treatment of stroke.
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