Preparation Technology and Determination of Annonaceous Acetogenin Dripping Pill
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Preparation Technology and Determination of Annonaceous Acetogenin Dripping Pill
Chinese Journal of Experimental Traditional Medical FormulaeVol. 18, Issue 1, Pages: 16-19(2012)
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Published:2012
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XU Sha-sha, LI Xiang, CHEN Jian-wei, et al. Preparation Technology and Determination of Annonaceous Acetogenin Dripping Pill[J]. Chinese journal of experimental traditional medical formulae, 2012, 18(1): 16-19.
DOI:
XU Sha-sha, LI Xiang, CHEN Jian-wei, et al. Preparation Technology and Determination of Annonaceous Acetogenin Dripping Pill[J]. Chinese journal of experimental traditional medical formulae, 2012, 18(1): 16-19.DOI:
Preparation Technology and Determination of Annonaceous Acetogenin Dripping Pill
Objective: To determine optimum preparation technology of annonaceous acetogenin dripping pill(AADP) by researching various factors on it. Method: Shape of dripping pill
hardness
dissolution time and pill weight as parameters to select formulation technology and dripping conditions of pill. The content of annonaceous total acetogenin was determined by UV spectrophotometry. Result: Optimum technology was: methyl-silicon oil as refrigerant
proportion of PEG4000-PEG6000 was 4 ∶1
annonaceous acetogenin to matrix was 1 ∶4
processing temperature was at 70 ℃
and cooling temperature was 5-15 ℃
dripping distance was 2 cm and ID/OD of emitter was 2/2.5 mm; The content of annonaceous total acetogenin was 2.53
2.54
2.66 mg. Conclusion: This process was simple
feasible and reproducible; Ultraviolet spectrophotometry method was simple
accurate and could be used to control quality of this dripping pill.
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